ut receptor — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T13272	UT-155		Androgen Receptor
	UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).		Androgen Receptor
T5171	Treprostinil Sodium	UT-15	VEGFR , c-RET , Prostaglandin Receptor
	Treprostinil Sodium (UT-15) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).		VEGFR , c-RET , Prostaglandin Receptor
T13273	UT-34		Androgen Receptor
	UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wild-type, F876L and W741L AR, respectively), and has anti-prost...		Androgen Receptor
T23323	SB 611812		Neurotensin Receptor
	SB 611812 is an antagonist of urotensin-II (UT) and can be used in studies about the treatment of cardiovascular disease.		Neurotensin Receptor
T2058	Palosuran	ACT-058362	GPR
	Palosuran (ACT-058362) (ACT-058362) is a new potent and specific antagonist of the human UT receptor.		GPR
T5150	Treprostinil	LRX-15,Orenitram,Remodulin	Prostaglandin Receptor
	Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).		Prostaglandin Receptor
TP1928L1	[Orn5]-URP acetate	[Orn5]-URP acetate(782485-03-4 free base)	GPR
	[Orn5]-URP acetate is an effective and selective Urotensin-II receptor (UT) antagonist (pEC50 = 7.24). [Orn5]-URP exhibits no agonist activity.		GPR
T22476	(±)-AC 7954 hydrochloride		Neurotensin Receptor
	(±)-AC 7954 hydrochloride is a urotensin-II (UT) receptor activator.		Neurotensin Receptor
TP2104L	UFP 803 acetate		Neurotensin Receptor
	UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.		Neurotensin Receptor
T4689	Palosuran hydrochloride 540769-28-6(free base）	ACT-058362 hydrochloride	GPR
	Palosuran hydrochloride 540769-28-6(free base)(ACT-058362 hydrochloride) is a new potent and specific antagonist of the human UT receptor with an IC50 of 3.6±0.2 nM.		GPR
T12848	SB-657510		Others , Neurotensin Receptor
	SB-657510 is a urotensin II (UII) receptor (UT) antagonist. The Ki values of UT for human, monkey, cat, rat and mouse were 61, 17, 30, 65 and 56 nM, respectively. SB-657510 plays an anti-inflammatory role by inhibiting U...		Others , Neurotensin Receptor
TP2106L	Urantide acetate(669089-53-6 free base)		Neurotensin Receptor
	Urantide acetate is a selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced ...		Neurotensin Receptor
T37527L	[Orn8]-Urotensin II acetate		GPR
	[Orn8]-Urotensin II acetate is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.		GPR
T13977	(R)-UT-155		Epigenetic Reader Domain
	(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.		Epigenetic Reader Domain
T23326	SB 706375		Others
	urotensin-II (UT) receptor antagonist		Others
T22815	GSK 1562590 hydrochloride		Others
	urotensin II (UT) receptor antagonist		Others
T75827	UFP-803 TFA
	UFP-803 TFA, a potent ligand for the urotensin-II receptor (UT), exhibits minimal residual agonist activity, rendering it a valuable asset for exploring the UT system's function in physiology and pathology [1].
T75828	[Orn5]-URP TFA
	[Orn5]-URP TFA acts as a potent and selective antagonist exclusively targeting the Urotensin-II receptor (UT), devoid of any agonist activity, and demonstrates a significant inhibitory efficiency with a pEC50 value of 7....
TP2106	Urantide
	Selective and competitive urotensin-II (UT) receptor antagonist (pKB = 8.3). Blocks hU-II induced contractions in thoracic aorta ex vivo. Exhibits no effect on noradrenaline or endothelin 1-induced contraction or on acet...
TP1928	[Orn5]-URP
	Urotensin-II (UT) receptor pure antagonist (pEC50 = 7.24). Displays no agonist activity unlike other U-II/URP analogs. Inhibits the action of U-II in the rat aorta ring assay.